Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK' and Ligand = 'BDBM50443180'
TargetTyrosine-protein kinase ITK/TSK(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443180(CHEMBL3086536)
Affinity DataKi:  0.700nMAssay Description:Inhibition of full length GST-tagged ITK (unknown origin) using Ac-EFPIYDFLPAKKK-NH2 as substrate after 35 mins by LC/MS analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50443180(CHEMBL3086536)
Affinity DataIC50:  91nMAssay Description:Inhibition of ITK in human Jurkat cells assessed as inhibition of PLC-gamma1 phosphorylation by immuno-detection assayMore data for this Ligand-Target Pair