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Found 4 Enz. Inhib. hit(s) with Target = 'UDP-N-acetylmuramoylalanine--D-glutamate ligase' and Ligand = 'BDBM50046818'
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.10E+4nMAssay Description:Competitive inhibition of Escherichia coli MurD using D-Glu substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.90E+4nMAssay Description:Partial non-competitive inhibition of Escherichia coli MurD using UMA substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  3.90E+4nMAssay Description:Partial un-competitive inhibition of Escherichia coli MurD using ATP substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed