Found 4 Enz. Inhib. hit(s) with Target = 'Ubiquitin carboxyl-terminal hydrolase 7' and Ligand = 'BDBM50560581'
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of recombinant full length USP7 (unknown origin) using di-ubiquitin as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.80E+5nMAssay Description:Allosteric binding affinity to USP7 catalytic domain (unknown origin) at Met328 residues by NMR-15N-1H TROSY spectral titration analysisMore data for this Ligand-Target Pair
Affinity DataKd: 5.40E+5nMAssay Description:Binding affinity to USP7 (unknown origin) by T2 relaxation experiment based analysisMore data for this Ligand-Target Pair
Affinity DataKd: 6.80E+5nMAssay Description:Allosteric binding affinity to USP7 catalytic domain (unknown origin) at Met328, Trp285, Gly284, Gln405 and Gly313 residues by NMR-15N-1H TROSY spect...More data for this Ligand-Target Pair