Found 6 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM35723' TargetVasopressin V1a receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
TargetVasopressin V1a receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 32nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 296nMAssay Description:Displacement of [3H]-vasopressin from human V1A receptor expressed in CHO cells membrane by microbeta scintillation counter analysisMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(RAT)
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
TargetVasopressin V1a receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 470nMAssay Description:Inhibition of human V1A receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescent plate readerMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 580nMpH: 7.4 T: 2°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
