Report error Found 15 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50065115'
Affinity DataIC50: 82nMAssay Description:In vitro inhibition of (Phe-3,4,5 [3H]-) AVP binding towards isolated rat hepatic Vasopressin V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of [3H]Arg-vasopressin binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Binding affinity towards human V1a receptorsMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]Arg-vasopressin from human recombinant vasopressin V1a receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against [3H]AVP binding to human vasopressin V1a receptor More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Displacement of [3H]AVP from vasopressin receptor (V1a) from human platelet membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of [3H]- AVP binding to V1a receptor from human platelet membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:In vitro binding affinity to human V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Displacement of (Phe-3,4,5-H) Vasopressin from V1a receptor from rat liver membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:In vitro binding affinity for rat V1a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of [3H]AVP binding to Dawley rat hepatic vasopressin V1a receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at human vasopressin V1a receptor expressed in HEK293 cells assessed as inhibition of Arg-vasopressin-induced intracellular calci...More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of 1 nM AVP-induced calcium mobilisation in cells expressing human vasopressin V1a receptorMore data for this Ligand-Target Pair
