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Found 2 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50114032'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114032(CHEMBL86577 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  3.03nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114032(CHEMBL86577 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  62.7nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed