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Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50152974'
TargetVasopressin V1a receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataKi:  196nMAssay Description:Displacement of DY647 from SNAP-tagged V1A receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human V1A receptor expressed in HEK cells assessed as inhibition of AVP-induced intracellular calcium flux incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed