Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50152974'
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50152974BDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human V1A receptor expressed in HEK cells assessed as inhibition of AVP-induced intracellular calcium flux incubated for 45 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50152974BDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataKi:  196nMAssay Description:Displacement of DY647 from SNAP-tagged V1A receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50152974BDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed