Found 2 Enz. Inhib. hit(s) with Target = 'Vesicular acetylcholine transporter' and Ligand = 'BDBM50018079'
Affinity DataKi: 40.6nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in rat PC12 cells after 60 minsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair