Found 4 Enz. Inhib. hit(s) with Target = 'Vesicular acetylcholine transporter' and Ligand = 'BDBM50292907'
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 cell membrane after 20 hrsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
Institute Of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Institute Of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Rattus norvegicus)
Institute Of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Institute Of Radiopharmaceutical Cancer Research
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair