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Found 3 Enz. Inhib. hit(s) with Target = 'Virokine/NFkB inhibitor' and Ligand = 'BDBM50316623'
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50316623((N,N)-N,N'-(1,2-bis(3,4,5-trimethoxyphenyl)ethane-...)
Affinity DataIC50:  2.40E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50316623((N,N)-N,N'-(1,2-bis(3,4,5-trimethoxyphenyl)ethane-...)
Affinity DataIC50:  2.40E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50316623((N,N)-N,N'-(1,2-bis(3,4,5-trimethoxyphenyl)ethane-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed