Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Vitamin D3 receptor' and Ligand = 'BDBM50135094'
TargetVitamin D3 receptor(Homo sapiens (Human))
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50135094(CHEMBL3745746)
Affinity DataIC50:  35nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from recombinant human VDR ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50135094(CHEMBL3745746)
Affinity DataEC50:  30nMAssay Description:Agonist activity at VDR in human HEK293 cells assessed as transcriptional activity after 16 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed