Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Vitamin D3 receptor' and Ligand = 'BDBM50455853'
TargetVitamin D3 receptor(Homo sapiens (Human))
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50455853(CHEMBL4202828)
Affinity DataIC50:  4.5nMAssay Description:Displacement of fluormone from human full length VDR after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50455853(CHEMBL4202828)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as increase in transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed