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Found 6 Enz. Inhib. hit(s) with Target = 'tRNA (guanine-N(1)-)-methyltransferase' and Ligand = 'BDBM50519349'
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50:  330nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50:  840nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  91nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  2.75E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  1.04E+4nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB