Affinity DataIC50: 14nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of CypD (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CypB (unknown origin)More data for this Ligand-Target Pair
TargetHeat shock factor protein 1(Homo sapiens (Human))
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair
TargetHeat shock factor protein 1(Homo sapiens (Human))
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of PPIL1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CypC (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CypB (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PPIL1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CypC (unknown origin)More data for this Ligand-Target Pair
TargetHeat shock factor protein 1(Homo sapiens (Human))
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair