Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity of the compound in radioreceptor binding assay by using [3H]-5-HT radioligand against 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Affinity DataKi: 20nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity in radioreceptor binding assay by using [3H]5-HT radioligand against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Albany Medical College
Curated by PDSP Ki Database
Albany Medical College
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Albany Medical College
Curated by PDSP Ki Database
Albany Medical College
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Binding affinity in radioreceptor binding assay by using [3H]5-HT radioligand against 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Binding affinity of the compound in radioreceptor binding assay by using [3H]-5-HT radioligand against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 116nMAssay Description:Intrinsic affinity of the compound towards serotonin receptor from rat frontal cortex by displacement of [3H]-5-HTMore data for this Ligand-Target Pair
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Albany Medical College
Curated by PDSP Ki Database
Albany Medical College
Curated by PDSP Ki Database
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortexMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Binding affinity to 5-hydroxytryptamine 2 receptor in rat frontal cortical membranes by [3H]- KET displacement.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Binding affinity of a compound to rat brain 5-hydroxytryptamine 1A (serotonin) receptor assayed by radiolabeled [3H]-8-OH-DPAT ligand displacementMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Evaluated for binding affinity towards 5-hydroxytryptamine 1A receptor in rat brainMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
National Institute of Neurological Disorders and Stroke
Curated by PDSP Ki Database
National Institute of Neurological Disorders and Stroke
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Albany Medical College
Curated by PDSP Ki Database
Albany Medical College
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 298nMAssay Description:Intrinsic affinity of the compound towards serotonin receptor from rat frontal cortex by displacement of [3H]-spiperone.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Albany Medical College
Curated by PDSP Ki Database
Albany Medical College
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Albany Medical College
Curated by PDSP Ki Database
Albany Medical College
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Alberta
Curated by PDSP Ki Database
University of Alberta
Curated by PDSP Ki Database
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 337nMAssay Description:Binding affinity against rat Alpha-1 adrenergic receptor.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University of Washington
Curated by PDSP Ki Database
University of Washington
Curated by PDSP Ki Database