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TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321827(4-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)-N,N...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317865(2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole |...)
Affinity DataEC50:  0.75nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321826(4-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)-N-m...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321816(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321824(4-((1H-Imidazol-4-yl)methyl)-1-(4-isopropylphenyl)...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321823(4-((1H-Imidazol-4-yl)methyl)-1-(3-(trifluoromethyl...)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321815(4-((1H-Imidazol-4-yl)methyl)-1-(4-(trifluoromethyl...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321822(4-((1H-Imidazol-4-yl)methyl)-1-(4-nitrophenyl)pipe...)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321821(4-((1H-Imidazol-4-yl)methyl)-1-(4-fluorophenyl)pip...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321820(4-((1H-Imidazol-4-yl)methyl)-1-phenylpiperidine | ...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321828(4-((1H-Imidazol-4-yl)methyl)-1-(naphthalen-2-yl)pi...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321829(3-(4-((1H-Imidazol-4-yl)methyl)piperidin-1-yl)pyri...)
Affinity DataEC50:  177nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM22542(4-(1H-imidazol-4-ylmethyl)piperidine | 4-(1H-imida...)
Affinity DataEC50:  0.670nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321825(4-((1H-Imidazol-4-yl)methyl)-1-(4-tert-butylphenyl...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed