Compile Data Set for Download or QSAR
Report error Found 9 of ki for UniProtKB: Q9H228
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559603BDBM50559603(CHEMBL4787458)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to recombinant human S1P5 receptor expressed in Chem-1 cell membrane by 33P-SIP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50250631BDBM50250631(CHEMBL4093489)
Affinity DataKi:  0.574nMAssay Description:Displacement of [33P]-S1P from human S1P5 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2019
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22202BDBM22202({[(4Z)-2-amino-3-hydroxyoctadec-4-en-1-yl]oxy}phos...)
Affinity DataKi:  0.920nM ΔG°:  -11.5kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559628BDBM50559628(CHEMBL4798593)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to recombinant human S1P5 receptor expressed in Chem-1 cell membrane by 33P-SIP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23165BDBM23165(CHEMBL366208 | [(2S)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataKi:  2.20nM ΔG°:  -11.0kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23163BDBM23163({2-amino-3-hydroxy-2-[2-(4-octylphenyl)ethyl]propo...)
Affinity DataKi:  4.20nM ΔG°:  -10.6kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559616BDBM50559616(CHEMBL4748198)
Affinity DataKi:  4.40nMAssay Description:Binding affinity to recombinant human S1P5 receptor expressed in Chem-1 cell membrane by 33P-SIP binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23164BDBM23164(CHEMBL190006 | [(2R)-2-amino-3-hydroxy-2-[2-(4-oct...)
Affinity DataKi:  121nM ΔG°:  -8.77kcal/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 5(Human)
Biogen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50494302BDBM50494302(CHEMBL3086532)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of S1P5 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed