Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at histamine H3 receptor in rat forebrain assessed as inhibition of [3H]histamine release from synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at histamine H3 receptor in rat forebrain assessed as inhibition of [3H]histamine release from synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Histamine-3 membranes were prepared from recombinant CHO-k1 cells expressing human histamine-3 receptor or rat histamine-3 receptor. Radioligand (RS)...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity at histamine H3 receptor in rat forebrain assessed as inhibition of [3H]histamine release from synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+3nMAssay Description:Displacement of [3H]SMT from histamine H3 receptor in forebrain of ratMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Antagonist activity at rat histamine H3 receptorMore data for this Ligand-Target Pair