Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of ic50 for UniProtKB: Q9BWU1
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50353060(CHEMBL4167193)
Affinity DataIC50:  8nMAssay Description:Inhibition of human CDK19 (M1 to N360 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50459995(CHEMBL4225966 | US11471446, Compound DBA-10)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50459995(CHEMBL4225966 | US11471446, Compound DBA-10)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50248631(CHEMBL4080906)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDK19 (unknown origin) in presence of [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM21079(1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50565105(CHEMBL4792974)
Affinity DataIC50:  29nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50540078(CHEMBL4639890)
Affinity DataIC50:  100nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  206nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50612439(CHEMBL5279425)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of GST-tagged human recombinant CDK11 (1 to 795 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50404389(CHEMBL5285499)
Affinity DataIC50: >1.20E+3nMAssay Description:Blocking activity against Beta-1 adrenergic receptor in spontaneously beating guinea pig atrial preparationsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50593922(CHEMBL5199065)
Affinity DataIC50: >1.20E+3nMAssay Description:Blocking activity against Beta-2 adrenergic receptor in guinea pig tracheal stripsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50539721(CHEMBL4635959)
Affinity DataIC50: >8.00E+3nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM62810(2-amino-6-methyl-4-(3-pyridinyl)-5,6,7,8-tetrahydr...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of CDK19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM62810(2-amino-6-methyl-4-(3-pyridinyl)-5,6,7,8-tetrahydr...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of recombinant CDK19 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed