TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.590nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.24nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.45nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 1.94nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]-Tyr4-bombesin from GRP receptor in human PC3 cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Displacement of [125I]-Tyr4-bombesin from GRP receptor in human PC3 cells after 1 hr by gamma-counting analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Antagonistic activity against labelled Bombesin receptor bb2 binding sites in rat cerebral cortex by using [125I]- [Tyr] bombesin in presence of NMB;...More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]-Tyr4-BBN from human GRPR overexpressed in human T47D cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Displacement of [125I]-Tyr4-bombesin from GRP receptor in human PC3 cells after 1 hr by gamma-counting analysisMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Binding affinity to GRP receptor (unknown origin)More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human GRP-R expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition gastrin-releasing peptide receptorMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]bombesin from human bombesin BB2 receptor expressed in NFAT-CHO cells after 2 hrs by liquid sci...More data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
National Center For Scientific Research Demokritos
Curated by ChEMBL
National Center For Scientific Research Demokritos
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human GRPRMore data for this Ligand-Target Pair