Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 182nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 366nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 366nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 387nMAssay Description:Displacement of [3H]clonidine from imidazoline 1 receptor in Sprague-Dawley rat kidneyMore data for this Ligand-Target Pair
Affinity DataIC50: 477nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 646nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 646nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 856nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.77E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.88E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.22E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.39E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 3.57E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.01E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.26E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.11E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.15E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 5.83E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.33E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of 3 nM [3H]-clonidine binding to rat kidney membrane imidazoline receptor I-1 in presence of rauwolscineMore data for this Ligand-Target Pair
Affinity DataIC50: 6.89E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7.24E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7.36E+3nMAssay Description:Displacement of [3H]clonidine from Imidazoline receptor 1 in Sprague-Dawley rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7.41E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 7.56E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.59E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Affinity DataIC50: 7.74E+3nMAssay Description:Displacement of [3H]2BF1 from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.75E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.78E+3nMAssay Description:Inhibition of Sprague-Dawley rat imidazoline I1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of 3 nM [3H]-clonidine binding to rat kidney membrane imidazoline receptor I-1 in presence of rauwolscineMore data for this Ligand-Target Pair