Affinity DataIC50: 0.0190nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Antagonism of the guinea pig tachykinin NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair