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Found 13 of ki for UniProtKB: P11474
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312096(4-bromo-6,8-dihydroxy-2-(4-hydroxyphenyl)isoquinol...)
Affinity DataKi:  32nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312133(US9604931, 12z)
Affinity DataKi:  40nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312140(6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...)
Affinity DataKi:  70nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312134(4-bromo-6-methoxy-2-(4-methoxyphenyl)-1-oxo-1,2-di...)
Affinity DataKi:  76nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312135(6,8-dihydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2-dihydr...)
Affinity DataKi:  94nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312151((E)-6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(prop-1-en...)
Affinity DataKi:  102nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312149(6,8-dihydroxy-2-(4-hydroxyphenyl)-4-(4-methoxyphen...)
Affinity DataKi:  124nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312139(2-(3-fluoro-4-hydroxyphenyl)-6,8-dihydroxy-4-vinyl...)
Affinity DataKi:  205nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312136(4-bromo-6-hydroxy-2-(4-hydroxyphenyl)-1-oxo-1,2-di...)
Affinity DataKi: >394nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM310198(4-bromo-6-hydroxy-2-(4-hydroxyphenyl)isoquinolin-1...)
Affinity DataKi:  998nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312137(6-hydroxy-2-(4-hydroxyphenyl)-4-phenylisoquinolin-...)
Affinity DataKi:  1.78E+3nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM312138(6-hydroxy-2-(4-hydroxyphenol)-4-(4-methoxyphenyl)i...)
Affinity DataKi:  2.10E+3nMAssay Description:Estrogen receptor (ERβ) binding affinity of the NRBAs was also determined using an in vitro competitive radioligand-binding assay with [3H]-estr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Gtx

US Patent
LigandPNGBDBM50091046(CHEMBL3582112)
Affinity DataKi: >2.30E+3nMAssay Description:Displacement of fluormone ES2 from human recombinant estrogen receptor-alpha expressed in insect Sf9 cells after 120 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed