Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ki data for polymerid = 50006416
TargetSphingosine kinase 1(Mus musculus)
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50041978(CHEMBL3134157)
Affinity DataKi:  3.60nMAssay Description:Inhibition of SphK1 in mouse erythrocytes using sphingosine as substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Mus musculus)
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50266437(CHEMBL4092871)
Affinity DataKi:  400nMAssay Description:Inhibition of recombinant mouse SPHK1 using sphingosine as substrate in presence ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Mus musculus)
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50407506(CHEMBL4595333)
Affinity DataKi: >2.00E+4nMAssay Description:Functional H2 receptor antagonistic activity in vitro assay on the isolated spontaneously beating guinea-pig right atriumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSphingosine kinase 1(Mus musculus)
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50407507(CHEMBL5281819)
Affinity DataKi:  2.00E+4nMAssay Description:Functional Histamine H3 receptor antagonistic activity in vitro assay on guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSphingosine kinase 1(Mus musculus)
Virginia Tech

Curated by ChEMBL
LigandPNGBDBM50514480(CHEMBL4466524)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of recombinant mouse SphK1 expressed in baculovirus infected Sf9 insect cells using D-erythro-sphingosine as substrate measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed