Compile Data Set for Download or QSAR
maximum 50k data
Found 25 of ic50 data for polymerid = 6607
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  52nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  93nMAssay Description:Inhibition of Influenza A virus (A/Shanghai/01/2014(H7N9)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271273(CHEMBL4127125)
Affinity DataIC50:  102nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  146nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50464877(CHEMBL4288789)
Affinity DataIC50:  166nMAssay Description:Inhibition of Influenza A virus (A/Shanghai/01/2014(H7N9)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271273(CHEMBL4127125)
Affinity DataIC50:  191nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  238nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50464876(CHEMBL4288995)
Affinity DataIC50:  426nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50181441(BCX-1812 | CHEBI:85202 | Peramivir)
Affinity DataIC50:  451nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase E119A mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271298(CHEMBL4128362)
Affinity DataIC50:  465nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50464877(CHEMBL4288789)
Affinity DataIC50:  564nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase E119A mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50464876(CHEMBL4288995)
Affinity DataIC50:  590nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase E119A mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50464877(CHEMBL4288789)
Affinity DataIC50:  640nMAssay Description:Inhibition of Influenza A virus (A/Vietnam/1194/2004 (H5N1)) recombinant neuraminidase R292K mutant expressed in HEK293 cells pre-incubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271265(CHEMBL4126987)
Affinity DataIC50:  3.68E+3nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271265(CHEMBL4126987)
Affinity DataIC50:  3.71E+3nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271264(CHEMBL4125754)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271264(CHEMBL4125754)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271266(CHEMBL4125895)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate preincubated for 60 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM139226(US8883846, 32)
Affinity DataKi:  5.00E+3nM ΔG°:  -7.23kcal/mole IC50:  3.00E+4nMT: 2°CAssay Description:Virus propagation: Influenza A/Brisbane/59/2007 (H1N1) virus was propagated in Madin-Darby Canine Kidney (MDCK) cells. Seed virus was inoculated into...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM50271266(CHEMBL4125895)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of Influenza A virus (A/Fukui/45/04(H3N2)) neuraminidase E119V mutant activity using 4-MUNANA as substrate measured every min for 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM139222(US8883846, 20 | US8883846, 31)
Affinity DataKi:  2.00E+4nM ΔG°:  -6.41kcal/mole IC50:  9.20E+4nMT: 2°CAssay Description:Virus propagation: Influenza A/Brisbane/59/2007 (H1N1) virus was propagated in Madin-Darby Canine Kidney (MDCK) cells. Seed virus was inoculated into...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM139224(US8883846, 27)
Affinity DataKi:  1.00E+6nM ΔG°:  -4.09kcal/mole IC50:  3.80E+6nMT: 2°CAssay Description:Virus propagation: Influenza A/Brisbane/59/2007 (H1N1) virus was propagated in Madin-Darby Canine Kidney (MDCK) cells. Seed virus was inoculated into...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM139222(US8883846, 20 | US8883846, 31)
Affinity DataIC50:  4.00E+6nMT: 2°CAssay Description:Virus propagation: Influenza A/Brisbane/59/2007 (H1N1) virus was propagated in Madin-Darby Canine Kidney (MDCK) cells. Seed virus was inoculated into...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNeuraminidase(Influenza A virus (A/Brisbane/59/2007(H1N1)))
Csiro Manufacturing

Curated by ChEMBL
LigandPNGBDBM139223(US8883846, 21)
Affinity DataIC50:  1.00E+7nMT: 2°CAssay Description:Virus propagation: Influenza A/Brisbane/59/2007 (H1N1) virus was propagated in Madin-Darby Canine Kidney (MDCK) cells. Seed virus was inoculated into...More data for this Ligand-Target Pair
In DepthDetails US Patent