TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Inhibition of mouse QPCT measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Effective concentration for antagonistic activity towards human progesterone in CV-1 cellsMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse glutaminyl cyclaseMore data for this Ligand-Target Pair
Ligand Info
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of mouse glutaminyl cyclase assessed as reduction in conversion of H-Gln-AMC hydrobromide to pGlu-AMC preincubated with substrate for 10 m...More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of mouse glutaminyl cyclaseMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of mouse glutaminyl cyclaseMore data for this Ligand-Target Pair
Ligand Info
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of mouse glutaminyl cyclaseMore data for this Ligand-Target Pair
Ligand Info
TargetGlutaminyl-peptide cyclotransferase(Mus musculus (mouse))
Seoul National University
Curated by ChEMBL
Seoul National University
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of mouse QPCT measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair