Compile Data Set for Download or QSAR
Found 10 of kd for UniProtKB: Q03181
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to human PPARdelta (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50192829(CHEMBL3958704 | US10188627, Compound 8a)
Affinity DataKd:  57nMAssay Description:Binding affinity to His-tagged PPARdelta (unknown origin) by SPR assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50085041(2-(4-(3-(4-acetyl-3-hydroxy-2-propylphenoxy)propox...)
Affinity DataKd:  76nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50122338((S)-3-[4-(3,3-Bis-biphenyl-4-yl-allyloxy)-phenyl]-...)
Affinity DataKd:  500nMAssay Description:Binding affinity towards peroxisome proliferator activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50428826(CHEMBL2337127)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to human PPARdelta (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50109547((S)-3-(4-(2-CARBAZOL-9-YL-ETHOXY)-PHENYL)-2-ETHOXY...)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity towards peroxisome proliferator activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50122340((S)-3-[4-(3,3-Diphenyl-allyloxy)-phenyl]-2-ethoxy-...)
Affinity DataKd:  5.70E+3nMAssay Description:Binding affinity towards peroxisome proliferator activated receptor deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50428827(CHEMBL2337126)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to human PPARdelta (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM91427(2-hydroxy-4-methoxy-3-(3-methylbut-2-enyl)-6-(2-ph...)
Affinity DataKd:  2.70E+4nMAssay Description:Binding affinity to human PPARdelta (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Helmholtz Centre for Infection Research

Curated by ChEMBL
LigandPNGBDBM50349826(SYRINGARESINOL)
Affinity DataKd:  2.76E+4nMAssay Description:Binding affinity to recombinant PPARbeta-LBD (254 to 441 residues) (unknown origin) expressed in Escherichia coli Rosetta2 cells by isothermal titrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed