Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 1251
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10406((1S,12S,14R)-4-[8-(1,3-dioxo-2,3-dihydro-1H-isoind...)
Affinity DataIC50:  10nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10417((1S,12S,14R)-4-[10-(1,3-dioxo-2,3-dihydro-1H-isoin...)
Affinity DataIC50:  20nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10415((1S,12S,14R)-4-[6-(1,3-dioxo-2,3-dihydro-1H-isoind...)
Affinity DataIC50:  40nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  50nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10430((1S,12S,14R)-9-{[10-(1,3-dioxo-2,3-dihydro-1H-isoi...)
Affinity DataIC50:  50nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10407((1S,12S,14R)-9-{[8-(1,3-dioxo-2,3-dihydro-1H-isoin...)
Affinity DataIC50:  70nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10423(10-N-Demethyl-10-N-(12 -trimethylammoniumdodecyl)g...)
Affinity DataIC50:  80nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10422(10-N-Demethyl-10-N-(10-trimethylammoniumdecyl) gal...)
Affinity DataIC50:  120nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10418((1S,12S,14R)-4-[12-(1,3-dioxo-2,3-dihydro-1H-isoin...)
Affinity DataIC50:  130nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10408((1S,12S,14R)-14-hydroxy-9-methoxy-4-methyl-11-oxa-...)
Affinity DataIC50:  140nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10405(2-{8-[(1S,12S,14R)-14-hydroxy-9-methoxy-11-oxa-4-a...)
Affinity DataIC50:  280nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10421(10-N-Demethyl-10-N-(8-trimethylammoniumoctyl) gala...)
Affinity DataIC50:  310nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10431((1S,12S,14R)-9-{[12-(1,3-dioxo-2,3-dihydro-1H-isoi...)
Affinity DataIC50:  320nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10412(10-N-Demethyl-10-N-(10-phthalimidodecyl)-galantham...)
Affinity DataIC50:  330nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  360nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10414((1S,12S,14R)-4-[4-(1,3-dioxo-2,3-dihydro-1H-isoind...)
Affinity DataIC50:  470nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10435(8-(Phthalimidooctyl)-trimethylammonium bromide | [...)
Affinity DataIC50:  900nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10410(10-N-Demethyl-10-N-(6-phthalimidohexyl)-galanthami...)
Affinity DataIC50:  990nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10434((12-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-az...)
Affinity DataIC50:  1.30E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10413(10-N-Demethyl-10-N-(12-phthalimidododecyl)-galanth...)
Affinity DataIC50:  1.40E+3nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10420(10-N-Demethyl-10-N-(6-trimethylammoniumhexyl) gala...)
Affinity DataIC50:  1.70E+3nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10409(10-N-Demethyl-10-N-(4-phthalimidobutyl)-galanthami...)
Affinity DataIC50:  2.00E+3nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10428((1S,12S,14R)-9-[4-(1,3-dioxo-2,3-dihydro-1H-isoind...)
Affinity DataIC50:  2.30E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10425(2-(8-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-a...)
Affinity DataIC50:  2.50E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10437(12-(Phthalimidododecyl)-trimethylammonium bromide ...)
Affinity DataIC50:  3.03E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10426(2-(10-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-...)
Affinity DataIC50:  4.00E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10433((10-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-az...)
Affinity DataIC50:  4.10E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10427(2-(12-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-...)
Affinity DataIC50:  4.60E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10436(10-(Phthalimidodecyl)-trimethylammonium bromide | ...)
Affinity DataIC50:  5.27E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10432((8-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-aza...)
Affinity DataIC50:  9.70E+3nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10419(10-N-Demethyl-10-N-(3-trimethylammoniumpropyl) gal...)
Affinity DataIC50:  1.24E+4nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Cnrs

LigandPNGBDBM10424(2-(4-{[(1S,12S,14R)-14-hydroxy-4-methyl-11-oxa-4-a...)
Affinity DataIC50:  1.61E+4nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed