Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 2327
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  1.20nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  1.40nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  25nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19463(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-propyl-3,4-dih...)
Affinity DataIC50:  29nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19469(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(2-methylpropy...)
Affinity DataIC50:  37nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19460((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methyl...)
Affinity DataIC50:  57nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19468(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methylbutyl...)
Affinity DataIC50:  59nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19460((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methyl...)
Affinity DataIC50:  68nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19465(8-Alkylnaringenin, 8d | 8-heptyl-5,7-dihydroxy-2-(...)
Affinity DataIC50:  69nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19469(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(2-methylpropy...)
Affinity DataIC50:  80nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19464(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-pentyl-3,4-dih...)
Affinity DataIC50:  97nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19466(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-nonyl-3,4-dihy...)
Affinity DataIC50:  113nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19468(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methylbutyl...)
Affinity DataIC50:  140nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19470(8-(2,2-dimethylpropyl)-5,7-dihydroxy-2-(4-hydroxyp...)
Affinity DataIC50:  141nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19463(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-propyl-3,4-dih...)
Affinity DataIC50:  155nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19470(8-(2,2-dimethylpropyl)-5,7-dihydroxy-2-(4-hydroxyp...)
Affinity DataIC50:  216nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19471(8-Alkylnaringenin, 8j | 8-benzyl-5,7-dihydroxy-2-(...)
Affinity DataIC50:  244nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19464(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-pentyl-3,4-dih...)
Affinity DataIC50:  383nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19465(8-Alkylnaringenin, 8d | 8-heptyl-5,7-dihydroxy-2-(...)
Affinity DataIC50:  392nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19467(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-undecyl-3,4-di...)
Affinity DataIC50:  421nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19466(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-nonyl-3,4-dihy...)
Affinity DataIC50:  436nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19471(8-Alkylnaringenin, 8j | 8-benzyl-5,7-dihydroxy-2-(...)
Affinity DataIC50:  503nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19462(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-methyl-3,4-dih...)
Affinity DataIC50:  863nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19467(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-undecyl-3,4-di...)
Affinity DataIC50:  1.02E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.15E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19462(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-methyl-3,4-dih...)
Affinity DataIC50:  5.25E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19461(α-CA inhibitor, 5 | 5,7-dihydroxy-2-(4-hydrox...)
Affinity DataIC50:  1.35E+4nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Ghent University

LigandPNGBDBM19461(α-CA inhibitor, 5 | 5,7-dihydroxy-2-(4-hydrox...)
Affinity DataIC50:  7.23E+4nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed