Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50048396
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214182(CHEMBL438929)
Affinity DataKi:  300nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214158(CHEMBL441586)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214157(CHEMBL411239)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214188(CHEMBL216870)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214188(CHEMBL216870)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214185(CHEMBL412507)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214155(CHEMBL413914)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50213962(CHEMBL410765)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214192(CHEMBL428833)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214193(CHEMBL410889)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214184(CHEMBL438420)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214173(CHEMBL442313)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214187(CHEMBL415828)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214156(CHEMBL414166)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214190(CHEMBL266910)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214160(CHEMBL436775)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214152(CHEMBL439107)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214178(CHEMBL439291)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214154(CHEMBL443593)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214159(CHEMBL415385)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214162(CHEMBL410689)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214180(CHEMBL415612)
Affinity DataKi:  5.50E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214189(CHEMBL266999)
Affinity DataKi:  5.50E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214179(CHEMBL411496)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214163(CHEMBL412745)
Affinity DataKi:  6.20E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214186(CHEMBL408320)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214183(CHEMBL264498)
Affinity DataKi:  1.07E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214151(CHEMBL414538)
Affinity DataKi:  1.20E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214191(CHEMBL269493)
Affinity DataKi:  1.55E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214174(CHEMBL411434)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214150(CHEMBL409378)
Affinity DataKi:  2.65E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214181(CHEMBL437667)
Affinity DataKi:  4.00E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50213963(CHEMBL410977)
Affinity DataKi:  7.50E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214176(CHEMBL262779)
Affinity DataKi:  8.90E+5nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214177(CHEMBL409189)
Affinity DataKi:  1.85E+6nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214153(CHEMBL216711)
Affinity DataKi:  2.05E+6nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214161(CHEMBL415172)
Affinity DataKi:  2.70E+6nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50214175(CHEMBL410027)
Affinity DataKi:  3.10E+6nMAssay Description:Inhibitory activity against interleukin-8 receptor using [125I]IL8More data for this Ligand-Target Pair
In DepthDetails
TargetC-X-C chemokine receptor type 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50213962(CHEMBL410765)
Affinity DataIC50:  1.90E+4nMAssay Description:Compound was tested for inhibitory activity against Interleukin-8 receptorMore data for this Ligand-Target Pair
In DepthDetails