Affinity DataKi: 1.22E+4nMAssay Description:Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 2.29E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 2.44E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.72E+4nMAssay Description:Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 4.75E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.07E+4nMAssay Description:Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 5.37E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 7.29E+4nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.12E+5nMAssay Description:Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+5nMAssay Description:Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 3.67E+5nMAssay Description:Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assayMore data for this Ligand-Target Pair