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Found 24 Enz. Inhib. hit(s) with all data for entry = 50035253
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108501(2-Methyl-furan-3-carboxylic acid (4-{5-[2-(4-dimet...)
Affinity DataKi:  0.102nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.620nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  1.20nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108493(2-Methyl-furan-3-carboxylic acid [4-({2-[4-([1,4']...)
Affinity DataKi:  2.90nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108494(2-Methyl-furan-3-carboxylic acid (4-{[2-(6-[1,4']b...)
Affinity DataKi:  5nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108495(1N-methyl-1N-{4-methyl-2-[6-(4-methylhexahydro-1-p...)
Affinity DataKi:  5.70nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108499(1N-methyl-1N-{4-methyl-2-[4-(4-methylhexahydro-1-p...)
Affinity DataKi:  7.60nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108500(2-Methyl-furan-3-carboxylic acid [4-(methyl-{4-met...)
Affinity DataKi:  8.80nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  24nMAssay Description:Evaluated for the binding affinity towards Vasopressin V1a receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108501(2-Methyl-furan-3-carboxylic acid (4-{5-[2-(4-dimet...)
Affinity DataKi:  34nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108493(2-Methyl-furan-3-carboxylic acid [4-({2-[4-([1,4']...)
Affinity DataKi:  42nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108500(2-Methyl-furan-3-carboxylic acid [4-(methyl-{4-met...)
Affinity DataKi:  73nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366798(CHEMBL1794053)
Affinity DataKi:  79nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108494(2-Methyl-furan-3-carboxylic acid (4-{[2-(6-[1,4']b...)
Affinity DataKi:  95nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366798(CHEMBL1794053)
Affinity DataKi:  168nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108497(2-Methyl-furan-3-carboxylic acid (4-{[4'-([1,4']bi...)
Affinity DataKi:  335nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108499(1N-methyl-1N-{4-methyl-2-[4-(4-methylhexahydro-1-p...)
Affinity DataKi:  445nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108502(2-Methyl-furan-3-carboxylic acid [4-({2-[3-([1,4']...)
Affinity DataKi:  491nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108495(1N-methyl-1N-{4-methyl-2-[6-(4-methylhexahydro-1-p...)
Affinity DataKi:  782nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108503(2-Methyl-furan-3-carboxylic acid [4-({2-[2-([1,4']...)
Affinity DataKi:  1.14E+3nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108502(2-Methyl-furan-3-carboxylic acid [4-({2-[3-([1,4']...)
Affinity DataKi:  1.36E+3nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108497(2-Methyl-furan-3-carboxylic acid (4-{[4'-([1,4']bi...)
Affinity DataKi:  2.04E+3nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108503(2-Methyl-furan-3-carboxylic acid [4-({2-[2-([1,4']...)
Affinity DataKi:  2.25E+3nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi: >1.00E+4nMAssay Description:Evaluated for the binding affinity towards Vasopressin V2 receptor in rat kidney membrane using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed