Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50036116
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.0100nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0120nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0130nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.0150nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  0.0160nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  0.0210nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  0.0230nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.0340nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  0.0360nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0870nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.110nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.240nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  4.20E+3nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi: >5.00E+3nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000554(3-[(2S,5R,8S,11R,14S)-14-(1H-Indol-3-ylmethyl)-11-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the porcine aortic smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000564(2-[2-{[2-(Cyclohexanecarbonyl-amino)-4-methyl-pent...)
Affinity DataIC50:  2.30E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000560(2-[2-({2-[(Azepane-1-carbonyl)-amino]-4-methyl-pen...)
Affinity DataIC50:  2.50E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000566((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50:  3.70E+3nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000559(2-(2-Azepan-1-yl-2-oxo-ethyl)-4-methyl-pentanoic a...)
Affinity DataIC50:  7.60E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000567(CHEMBL287980 | Sodium; ({2-[2-({2-[(azepane-1-carb...)
Affinity DataIC50:  7.60E+3nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000563(3-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionyl...)
Affinity DataIC50:  1.30E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000561(CHEMBL290454 | Sodium; 2-{2-[2-({2-[(azepane-1-car...)
Affinity DataIC50:  2.10E+4nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataIC50:  2.20E+4nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the porcine aortic smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataIC50:  2.30E+4nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the porcine cerebellum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000568(2-[2-({2-[2-(2-Chloro-phenyl)-acetylamino]-4-methy...)
Affinity DataIC50:  3.20E+4nMAssay Description:Compound was evaluated for the binding affinity towards Endothelin A receptor in porcine aortic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000565((S)-3-{(S)-2-[(S)-2-Amino-3-(3H-imidazol-4-yl)-pro...)
Affinity DataIC50:  4.40E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000553((S)-3-{(S)-2-[(S)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50:  5.80E+4nMAssay Description:Compound was evaluated for the binding affinity to endothelin receptor in the rat heart ventricle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000554(3-[(2S,5R,8S,11R,14S)-14-(1H-Indol-3-ylmethyl)-11-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the porcine cerebellum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B/1 receptor(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000564(2-[2-{[2-(Cyclohexanecarbonyl-amino)-4-methyl-pent...)
Affinity DataIC50:  2.30E+5nMAssay Description:Compound was evaluated for the binding affinity to Endothelin A receptor in the rat atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed