Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50043389
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50310892(CHEMBL1078511 | N,N'-(9-(2-(1-methylpyrrolidin-2-y...)
Affinity DataIC50:  18nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440391(CHEMBL2425367)
Affinity DataIC50:  28nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50134018(CHEMBL335819 | N,N'-(9-(4-aminophenylamino)acridin...)
Affinity DataIC50:  60nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440390(ISOMETAMIDIUM)
Affinity DataIC50:  100nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440389(CHEMBL1997011)
Affinity DataIC50:  100nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440388(CHEMBL2425366)
Affinity DataIC50:  130nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440387(CHEMBL2425365)
Affinity DataIC50:  220nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50176906(CHEMBL219728 | N'-(10H-indolo[3,2-b]quinolin-11-yl...)
Affinity DataIC50:  440nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50111322(CHEMBL274335 | N,N-Dimethyl-N'-(11-nitro-13H-5,13-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440386(CHEMBL2425364)
Affinity DataIC50:  750nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440385(CHEMBL2425363)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50068304(CHEMBL343445 | N-[9,10-Dioxo-6-(3-pyrrolidin-1-yl-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440384(CHEMBL2425362)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412201(CRYPTOLEPINE HYDROCHLORIDE | Cryptolepine)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440382(CHEMBL2425361)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440381(MERIDINE)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed