Affinity DataKi: 13nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor in mouse whole brain membrane measured after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 153nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 574nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 714nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 828nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 897nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.46E+3nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.87E+3nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor in mouse spleen membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.94E+3nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in HEK293-EBNA cell membranes after 90 mins by scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Displacement of [3H]-CP55940 from recombinant CB2 receptor (unknown origin) expressed in cell membranes after 90 mins by scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 6.21E+3nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in HEK293-EBNA cell membranes after 90 mins by scintillation counting meth...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataKi: 6.73E+3nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor in rat spleen membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor in mouse spleen membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 8.38E+3nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor in mouse spleen membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 9.04E+3nMAssay Description:Displacement of [3H]-CP55940 from recombinant CB2 receptor (unknown origin) expressed in cell membranes after 90 mins by scintillation counting metho...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor in rat spleen membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.47E+4nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in Sf9 cell membranes co-expressing Galphai3beta1gamma2 measured after 90 ...More data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor measured after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataKi: 2.46E+4nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor in rat spleen membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.36E+4nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.57E+4nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.83E+4nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor measured after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB2 receptor expressed in HEK293 cell membranes after 90 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from recombinant human CB1 receptor expressed in HEK293-EBNA cell membranes after 90 mins by scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 4.28E+4nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.73E+4nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 9.56E+4nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of MAGL in human U937 cell homogenates using [3H]-2OG as substrate preincubated for 15 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetFatty acid-binding protein 5(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of NBD-Stearate from recombinant human FABP5 measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.61E+5nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of recombinant human FAAH using N-arachidonyl-7-amino-4-methylcoumarin as substrate preincubated for 20 mins followed by substrate additio...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of recombinant human FAAH using N-arachidonyl-7-amino-4-methylcoumarin as substrate preincubated for 20 mins followed by substrate additio...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human FAAH using N-arachidonyl-7-amino-4-methylcoumarin as substrate preincubated for 20 mins followed by substrate additio...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of recombinant human FAAH using N-arachidonyl-7-amino-4-methylcoumarin as substrate preincubated for 20 mins followed by substrate additio...More data for this Ligand-Target Pair
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by b...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of recombinant human FAAH using N-arachidonyl-7-amino-4-methylcoumarin as substrate preincubated for 20 mins followed by substrate additio...More data for this Ligand-Target Pair
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by b...More data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of recombinant human NAAA expressed in HEK293 cells using [14C]-N-palmitoylethanolamine as substrate measured after 30 mins by beta-counti...More data for this Ligand-Target Pair
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by b...More data for this Ligand-Target Pair
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 3.05E+4nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by b...More data for this Ligand-Target Pair
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by b...More data for this Ligand-Target Pair