Found 94 Enz. Inhib. hit(s) with all data for entry = 50013370 
Affinity DataKi: 0.0270nMAssay Description:Displacement of [125I]EYF from human NPFFR2 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-FFRF-NH2 from human NPFFR1 expressed in CHO cell membrane by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of TAMRA-NPFF from human NPFFR2 expressed in CHO-K1 cells preincubated for 15 mins followed by GTPgammaS addition and measured after 15 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]-1DMeNPFF from rat NPFFR1 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]-1DMeNPFF from rat NPFFR2 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of TAMRA-NPFF from human NPFFR2 expressed in CHO-K1 cells preincubated for 15 mins followed by GTPgammaS addition and measured after 15 ...More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [125I]-1DMeNPFF from human NPFFR2 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [125I]EYF from human NPFFR2 expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to rat NPFFR1 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of [125I]-1DMeNPFF from human NPFFR1 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human NPFFR1 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [125I]EYF from human NPFFR2 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human NPFFR1 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to rat NPFFR1 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]-1DMeNPFF from human NPFFR2 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]-1DMeNPFF from rat NPFFR1 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]-1DMeNPFF from rat NPFFR2 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-FFRF-NH2 from human NPFFR2 expressed in CHO cell membrane by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [125I]-1DMeNPFF from human NPFFR1 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [125I]Tyr-NPFF from human NPFFR2 expressed in green monkey Cos-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Binding affinity to human NPFFR2 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of 125I-NPFF from human NPFFR1 incubated for 2 hrs by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [125I](Tyr)NPF from rat NPFFR1 expressed in rat PC12 cells incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Binding affinity to human NPFFR2 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of 125I-NPFF from human NPFFR2 incubated for 2 hrs by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 172nMAssay Description:Displacement of [3H]-FFRF-NH2 from human FLAG-tagged NPFFR1 expressed in CHO cell membrane incubated for 30 mins by Topcount scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:Binding affinity to rat NPFFR2 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 282nMAssay Description:Binding affinity to rat NPFFR2 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 461nMAssay Description:Displacement of [125I]Tyr-NPFF from human NPFFR2 expressed in green monkey Cos-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Displacement of [3H]-FFRF-NH2 from human FLAG-tagged NPFFR2 expressed in CHO cell membrane incubated for 30 mins by Topcount scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Displacement of [125I]NPFF from human NPFFR1 expressed in CHO cell membranes incubated for 120 mins by scintillation/luminescence counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 890nMAssay Description:Displacement of [125I]NPFF from human NPFFR1 expressed in CHO cell membranes incubated for 120 mins by scintillation/luminescence counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.44E+3nMAssay Description:Displacement of [125I]NPFF from human NPFFR2 expressed in CHO cell membranes incubated for 120 mins by scintillation/luminescence counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+3nMAssay Description:Displacement of [125I]NPFF from human NPFFR2 expressed in CHO cell membranes incubated for 120 mins by scintillation/luminescence counting methodMore data for this Ligand-Target Pair
TargetProlactin-releasing peptide receptor(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-PrRP-20 from human PrRP receptor expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
TargetProlactin-releasing peptide receptor(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-PrRP-20 from human PrRP receptor expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-Kp-10 from human KISS1R expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]-Kp-10 from human KISS1R expressed in CHO cell membrane by TopCount scintillation counter methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I](Tyr)NPF from rat NPFFR1 expressed in rat PC12 cells incubated for 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human NPFFR1 expressed in CHO-K1 cells assessed as reversal of agonist-induced inhibition of forskolin-stimulated cAMP accumul...More data for this Ligand-Target Pair
Affinity DataIC50: 387nMAssay Description:Antagonist activity at human NPFFR2 expressed in CHO-K1 cells assessed as reversal of agonist-induced inhibition of forskolin-stimulated cAMP accumul...More data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) expressed in HEK-293A cells assessed as inhibition of forskolin-induced cAMP accumulation ...More data for this Ligand-Target Pair
