Compile Data Set for Download or QSAR
maximum 50k data
Found 227 Enz. Inhib. hit(s) with all data for entry = 50019105
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321424(6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-...)
Affinity DataIC50:  5nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321411(6-[(E)-but-2-enyl]-4-[3-methoxy-4-(morpholine-4-ca...)
Affinity DataIC50:  6nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321412(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)
Affinity DataIC50:  7nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321422(5-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)
Affinity DataIC50:  8nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321437((E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-...)
Affinity DataIC50:  8nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321415(6-[(E)-but-2-enyl]-2-methyl-4-[3-methyl-4-(morphol...)
Affinity DataIC50:  9nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321407(6-[(E)-but-2-enyl]-2-methyl-4-[4-(morpholine-4-car...)
Affinity DataIC50:  12nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataIC50:  31nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataIC50:  48nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM321402(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)
Affinity DataIC50:  53nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))TBA
LigandPNGBDBM50532326(CHEMBL4519632)
Affinity DataIC50:  160nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD9 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321422(5-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)
Affinity DataIC50:  370nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM50532326(CHEMBL4519632)
Affinity DataIC50:  410nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321412(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)
Affinity DataIC50:  460nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50532326(CHEMBL4519632)
Affinity DataIC50:  460nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM321422(5-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)
Affinity DataIC50:  520nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM321407(6-[(E)-but-2-enyl]-2-methyl-4-[4-(morpholine-4-car...)
Affinity DataIC50:  750nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321407(6-[(E)-but-2-enyl]-2-methyl-4-[4-(morpholine-4-car...)
Affinity DataIC50:  810nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321411(6-[(E)-but-2-enyl]-4-[3-methoxy-4-(morpholine-4-ca...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321415(6-[(E)-but-2-enyl]-2-methyl-4-[3-methyl-4-(morphol...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50532326(CHEMBL4519632)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM321412(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321407(6-[(E)-but-2-enyl]-2-methyl-4-[4-(morpholine-4-car...)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM321411(6-[(E)-but-2-enyl]-4-[3-methoxy-4-(morpholine-4-ca...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321424(6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-...)
Affinity DataIC50:  2.40E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM321415(6-[(E)-but-2-enyl]-2-methyl-4-[3-methyl-4-(morphol...)
Affinity DataIC50:  2.80E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321402(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)
Affinity DataIC50:  3.30E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321411(6-[(E)-but-2-enyl]-4-[3-methoxy-4-(morpholine-4-ca...)
Affinity DataIC50:  3.30E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataIC50:  3.40E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321412(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)
Affinity DataIC50:  3.50E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human GABA-B receptor at 10 uM relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321422(5-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)
Affinity DataIC50:  4.20E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321437((E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-...)
Affinity DataIC50:  4.30E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))TBA
LigandPNGBDBM321402(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)
Affinity DataIC50:  4.70E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged CECR2 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataIC50:  5.10E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM321402(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50532326(CHEMBL4519632)
Affinity DataIC50:  5.70E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321415(6-[(E)-but-2-enyl]-2-methyl-4-[3-methyl-4-(morphol...)
Affinity DataIC50:  6.00E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321402(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)
Affinity DataIC50:  6.10E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321407(6-[(E)-but-2-enyl]-2-methyl-4-[4-(morpholine-4-car...)
Affinity DataIC50:  6.70E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataIC50:  8.30E+3nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetStromelysin-3(Mus musculus)TBA
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataIC50:  1.02E+4nMAssay Description:Cytotoxicity against human NB1 cells measured after 8 daysMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321412(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)
Affinity DataIC50:  1.23E+4nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321422(5-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)
Affinity DataIC50:  1.35E+4nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321415(6-[(E)-but-2-enyl]-2-methyl-4-[3-methyl-4-(morphol...)
Affinity DataIC50:  1.44E+4nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM321411(6-[(E)-but-2-enyl]-4-[3-methoxy-4-(morpholine-4-ca...)
Affinity DataIC50:  1.74E+4nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged BRD4 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetStromelysin-3(Mus musculus)TBA
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataIC50:  2.00E+4nMAssay Description:Cytotoxicity against human NB1 cells measured after 8 daysMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataIC50: >2.00E+4nMAssay Description:Displacement of biotinylated small-molecule ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 227 total ) | Next | Last >>
Jump to: