Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50046845
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134198(CHEMBL1684609)
Affinity DataIC50:  690nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin) expressed in CHO-K1 cells assessed as inhibition of trypsin-induced calcium flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134197(CHEMBL3735493)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin) expressed in CHO-K1 cells assessed as inhibition of trypsin-induced calcium flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134196(CHEMBL3736126)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin) expressed in CHO-K1 cells assessed as inhibition of trypsin-induced calcium flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed