Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50009967
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Affinity DataKi:  16nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533828(CHEMBL4570031)
Affinity DataKi:  184nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533823(CHEMBL494210)
Affinity DataKi:  5.04E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533825(CHEMBL4460819)
Affinity DataKi:  5.44E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533832(CHEMBL4524434)
Affinity DataKi:  5.64E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533830(CHEMBL4460655)
Affinity DataKi:  8.56E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533829(CHEMBL4592393)
Affinity DataKi:  8.75E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533827(CHEMBL4457103)
Affinity DataKi:  9.18E+3nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533833(CHEMBL4545415)
Affinity DataKi:  1.11E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533831(CHEMBL4445820)
Affinity DataKi:  1.51E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533834(CHEMBL4448716)
Affinity DataKi:  1.95E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533824(CHEMBL4574016)
Affinity DataKi:  2.52E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50533826(CHEMBL4520524)
Affinity DataKi:  2.54E+4nMAssay Description:Reversible inhibition of recombinant human Adk-short expressed in Escherichia coli BL21[DE3] assessed as [3H]AMP formation preincubated for 15 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed