TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Upr 2301, Cnrs
Curated by ChEMBL
Upr 2301, Cnrs
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein c...More data for this Ligand-Target Pair