Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50010040
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50534550(CHEMBL4542697)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human muscarinic M4 receptor assessed as inhibition of acetylcholine-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50534551(CHEMBL4448840)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human muscarinic M4 receptor assessed as inhibition of acetylcholine-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50042441(CHEMBL3353290)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human muscarinic M4 receptor assessed as inhibition of acetylcholine-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50445222(CHEMBL3105228)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human muscarinic M4 receptor assessed as inhibition of acetylcholine-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed