Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 50035212
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50099313(((3S,4R)-1-Methyl-4-phenyl-pyrrolidin-3-yl)-pyridi...)
Affinity DataIC50:  494nMAssay Description:Functional cocaine antagonism was evaluated by inhibition of [3H]dopamine reuptake at a concentration of 300 nM with cocaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50099304(CHEMBL275541 | [(3S,4R)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataIC50:  641nMAssay Description:Functional cocaine antagonism was evaluated by inhibition of [3H]dopamine reuptake at a concentration of 100 nM with cocaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed