Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50015470
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Goethe-University

Curated by ChEMBL
LigandPNGBDBM50586970(CHEMBL5074383)
Affinity DataIC50:  650nMAssay Description:Partial agonist activity at recombinant sGSF-PPARgamma (unknown origin) assessed as reduction in rosiglitazone induced CBP-1 recruitment incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Goethe-University

Curated by ChEMBL
LigandPNGBDBM50586956(CHEMBL5075652)
Affinity DataIC50:  840nMAssay Description:Partial agonist activity at recombinant sGSF-PPARgamma (unknown origin) assessed as reduction in rosiglitazone induced CBP-1 recruitment incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Goethe-University

Curated by ChEMBL
LigandPNGBDBM50586944(CHEMBL5090821)
Affinity DataIC50:  1.62E+3nMAssay Description:Partial agonist activity at recombinant sGSF-PPARgamma (unknown origin) assessed as reduction in rosiglitazone induced CBP-1 recruitment incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed