Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with all data for assayid = 6 entry = 50039243
TargetPeroxisome proliferator-activated receptor gamma(Rattus norvegicus)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50322695(4,6-Bis(benzylthio)-2-(methylthio)pyrimidine-5-car...)
Affinity DataIC50:  539nMAssay Description:Antagonist activity at rat PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced luciferas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed