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TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86694(N'-(3-Chloro-4-morpholinophenyl)-N-hydroxyform...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  6nMAssay Description:Compound was evaluated in vitro for inhibition of Prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50172479((S)-FLURBIPROFEN | CHEMBL435298)
Affinity DataIC50:  30nMAssay Description:Concentration required to inhibit cyclooxygenase-1 in rat bloodMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286821(2-(2-Ethyl-10H-9-oxa-1-aza-anthracen-6-yl)-propion...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against COX-1 from rat peritoneal leukocytes, measured by PGE-2 produced (enzyme immunoassay)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50074922((+-)-2-fluoro-alpha-methyl-4-biphenylacetic acid |...)
Affinity DataIC50:  170nMAssay Description:Concentration required to inhibit cyclooxygenase-1 in rat bloodMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286822(2-(2-Methyl-10H-9-oxa-1-aza-anthracen-6-yl)-propio...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity of the compound against COX-1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105293(2-(4-Benzyl-7-methoxy-naphthalen-1-yl)-propionic a...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50012860(1-Oxo-1,2-dihydro-6-oxa-10b-aza-aceanthrylene-2-ca...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of cyclooxygenase-1 in rat RBL-1 cells preincubated for 10 mins followed by [14C]arachidonic acid addition and measured after 5 mins by ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105289(2-[4-(4-Fluoro-benzyl)-7-methoxy-naphthalen-1-yl]-...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105298(2-[4-(2-Chloro-benzyl)-7-methoxy-naphthalen-1-yl]-...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105284(2-[4-(4-Fluoro-benzyl)-naphthalen-1-yl]-propionic ...)
Affinity DataIC50:  2.40E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105290(2-[7-Methoxy-4-(4-methyl-benzyl)-naphthalen-1-yl]-...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286819(CHEMBL367463 | Pranoprofen | i2-(10H-9-Oxa-1-aza-a...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory activity of the compound against COX-1 from ram seminal vesiclesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105303(2-[4-(4-Chloro-benzyl)-7-methoxy-naphthalen-1-yl]-...)
Affinity DataIC50:  4.10E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105286(2-[4-(4-Fluoro-benzyl)-7-methoxy-naphthalen-1-yl]-...)
Affinity DataIC50:  7.30E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105302(2-[7-Methoxy-4-(4-methoxy-benzyl)-naphthalen-1-yl]...)
Affinity DataIC50:  8.80E+3nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289091((S)-4-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-in...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated in vitro for inhibition of Prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289090(CHEMBL162776 | {1-[1-(4-Bromo-benzyl)-5-methoxy-2-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289087(4-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289088(4-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289087(4-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated in vitro for inhibition of Prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289092((R)-4-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-in...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated in vitro for inhibition of Prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289089(2-[1-(4-Chloro-benzyl)-5-methoxy-2-methyl-1H-indol...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22369(4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofu...)
Affinity DataIC50:  1.14E+4nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.42E+4nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105285(2-[4-(4-Chloro-benzyl)-7-methylsulfanyl-naphthalen...)
Affinity DataIC50:  1.99E+4nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013686(CHEMBL3264520)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013687(CHEMBL3264523)
Affinity DataIC50:  2.79E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013684(CHEMBL3264519)
Affinity DataIC50:  2.98E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of COX-1 in rat peritoneal macrophages assessed as reduction in [125I]-6-Keto-PGF1alpha production using arachidonic acid as substrate pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013679(CHEMBL3264514)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013680(CHEMBL3264515)
Affinity DataIC50:  3.58E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105294(2-[4-(4-Fluoro-benzyl)-7-methoxy-naphthalen-1-yl]-...)
Affinity DataIC50:  3.58E+4nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013682(CHEMBL3264517)
Affinity DataIC50:  3.81E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50105301(2-[4-(4-tert-Butyl-benzyl)-7-methoxy-naphthalen-1-...)
Affinity DataIC50:  4.08E+4nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22970(2-{1-[(4-bromophenyl)methyl]-5-methoxy-2-methyl-1H...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013683(CHEMBL3264518)
Affinity DataIC50:  4.25E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50172473((-)-(2R)-2-(2-fluorobiphenyl-4-yl)propanoic acid |...)
Affinity DataIC50:  4.40E+4nMAssay Description:Concentration required to inhibit cyclooxygenase-1 in rat bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013688(CHEMBL3264524)
Affinity DataIC50:  4.75E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50260464(CHEMBL4071383)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of COX-1 in rat peritoneal macrophages assessed as reduction in [125I]-6-Keto-PGF1alpha production using arachidonic acid as substrate pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013681(CHEMBL3264516)
Affinity DataIC50:  4.97E+4nMAssay Description:Inhibition of rat seminal vesicle COX-1 using arachidonic acid as substrate assessed as reduction of PGG2 to PGH2 incubated for 1 min prior to substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289084(3-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50260465(CHEMBL4101003)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of COX-1 in rat peritoneal macrophages assessed as reduction in [125I]-6-Keto-PGF1alpha production using arachidonic acid as substrate pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289082(3-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289086((2R,3S)-3-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50289083(3-[1-(4-Bromo-benzyl)-5-methoxy-2-methyl-1H-indol-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Prostaglandin G/H synthase 1 using whole cell assayMore data for this Ligand-Target Pair
In DepthDetails Article
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