TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Competitive inhibition of porcine liver carboxylesterase by double reciprocal Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Inhibition of pig liver carboxylesterase by Lineweaver-Burk analysisMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 337nMAssay Description:Competitive inhibition of porcine liver carboxylesterase by double reciprocal Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 570nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.09E+3nMAssay Description:Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.33E+3nMAssay Description:Inhibition of pig liver carboxylesterase by Lineweaver-Burk analysisMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.54E+3nMAssay Description:Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 6.51E+3nMAssay Description:Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 6.64E+3nMAssay Description:Inhibition of pig liver carboxylesterase by Lineweaver-Burk analysisMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 7.37E+3nMAssay Description:Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 7.81E+3nMAssay Description:Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 0.457nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.32nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 9.30nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 10.5nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 17.0nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Institute Of Physiologically Active Compounds Russian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of Sus scrofa (pig) carboxylesterase isolated from liver in using p-nitrophenyl acetate as substrate incubated for 5 min prior to substrat...More data for this Ligand-Target Pair