Compile Data Set for Download or QSAR
maximum 50k data
Found 6
TargetProprotein convertase subtilisin/kexin type 6(Rattus norvegicus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270054(CHEMBL502642 | TPRARRRKKRT)
Affinity DataKi:  162nMAssay Description:Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Rattus norvegicus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270067(CHEMBL503520 | TPQRARRRKKRW)
Affinity DataKi:  192nMAssay Description:Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Rattus norvegicus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50269901(CHEMBL525748 | TPRARRRKKRI)
Affinity DataKi:  267nMAssay Description:Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Rattus norvegicus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270060(CHEMBL455792 | TPQRARRRKKRT)
Affinity DataKi:  296nMAssay Description:Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Rattus norvegicus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270068(CHEMBL500184 | TPQRARRRKKRF)
Affinity DataKi:  602nMAssay Description:Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Rattus norvegicus)
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50270069(CHEMBL499438 | TPQRARRRKKRY)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed