Compile Data Set for Download or QSAR
maximum 50k data
Found 63 of ec50 data for polymerid = 10753,49000313
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295697(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  1.78E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295696(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  3.08E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295695(2-(3-aminopropoxy)-N-(4-(3-aminopropoxy)benzyl)-N-...)
Affinity DataEC50:  3.18E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295695(2-(3-aminopropoxy)-N-(4-(3-aminopropoxy)benzyl)-N-...)
Affinity DataEC50:  5.40E+3nMAssay Description:Displacement of [125I]GVIA from rat brain membrane Cav2.2 after 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295697(2-(3-aminopropoxy)-N-(4-(3-(diaminomethyleneamino)...)
Affinity DataEC50:  5.70E+3nMAssay Description:Displacement of [125I]GVIA from rat brain membrane Cav2.2 after 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295701(CHEMBL565078 | N-(3-{4-[(6-Phenoxy-benzothiazol-2-...)
Affinity DataEC50:  5.80E+3nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304189(CHEMBL593380 | N-(4-(4-Fluorophenoxy)phenyl)-2-(8-...)
Affinity DataEC50:  6.00E+3nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400564(CHEMBL2206242)
Affinity DataEC50:  7.21E+3nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400566(CHEMBL2206239)
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295707(2-(3-(4-((2,2-diphenylethylamino)methyl)phenoxy)pr...)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304185(2-(5-Guanidino-octanamido)-5-(3-guanidinopropoxy)-...)
Affinity DataEC50:  1.30E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400565(CHEMBL2206262)
Affinity DataEC50:  1.42E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304187(2-(5-Guanidino-octanamido)-5-(3-guanidinobutoxy)-N...)
Affinity DataEC50:  1.50E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304188(2-(8-Guanidinooctanamido)-5-(3-guanidinopropoxy)-N...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304184(2-(5-Guanidinohexanamido)-5-(3-guanidinopropoxy)-N...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304186(2-(5-Guanidinohexanamido)-5-(3-guanidinobutoxy)-N-...)
Affinity DataEC50:  1.70E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295703(2-(3-(4-((4-phenoxyphenylamino)methyl)phenoxy)prop...)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295705(2-(3-(4-((benzhydrylamino)methyl)phenoxy)propyl)gu...)
Affinity DataEC50:  2.30E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataEC50:  2.76E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400563(CHEMBL2206241)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295699(2-(3-Guanidino-propoxy)-N-(6-phenoxy-benzothiazol-...)
Affinity DataEC50:  3.30E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295702(CHEMBL552193 | [4-(3-Amino-propoxy)-benzyl]-(4-phe...)
Affinity DataEC50:  3.40E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400567(CHEMBL2206248)
Affinity DataEC50: >7.00E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304180(2-(8-Aminooctanamido)-5-(3-aminopropoxy)-N-(4-phen...)
Affinity DataEC50:  7.20E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295700(CHEMBL550448 | [4-(3-Amino-propoxy)-benzyl]-(6-phe...)
Affinity DataEC50:  7.60E+4nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304190(2-(5-Aminopentanamido)-5-(3-aminopropoxy)-N-(4-phe...)
Affinity DataEC50:  7.70E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366800(OLOMOUCINE II)
Affinity DataEC50:  8.00E+4nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304182(5-(4-Aminobutoxy)-2-(8-aminooctanamido)-N-(4-pheno...)
Affinity DataEC50:  9.00E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50304181(5-(4-Aminobutoxy)-2-(6-aminohexanamido)-N-(4-pheno...)
Affinity DataEC50:  9.90E+4nMAssay Description:Displacement of [125I]GVIA from Cav2.2 channel in rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400584(CHEMBL2206259)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400578(CHEMBL2206245)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400582(CHEMBL2206261)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400581(CHEMBL2206263)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295698(2-(3-Amino-propoxy)-N-(6-phenoxy-benzothiazol-2-yl...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295704(3-{4-[(Benzhydryl-amino)-methyl]-phenoxy}-propylam...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400580(CHEMBL2206243)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400583(CHEMBL2206260)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400579(CHEMBL2206244)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Rattus norvegicus (Rat))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50295706(3-{4-[(2,2-Diphenyl-ethylamino)-methyl]-phenoxy}-p...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rat neuronal Cav2.2 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400568(CHEMBL2206240)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400569(CHEMBL2206255)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50378235(CHEMBL461557)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50358220(CHEMBL455389)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400570(CHEMBL2206254)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400571(CHEMBL2206253)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400572(CHEMBL2206252)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400573(CHEMBL2206251)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400574(CHEMBL2206250)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400575(CHEMBL2206249)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400576(CHEMBL2206247)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at N-type Cav2.2 channel expressed in tsA201 cell assessed as calcium current by whole-cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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