Affinity DataEC50: 3.30nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 6.40nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 11.2nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 12.8nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 17.6nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Inhibition of human DNA topoisomerase 1-mediated DNA cleavage assessed as relaxation of supercoiled pBR322 plasmid DNA after 15 mins by densitometerMore data for this Ligand-Target Pair
Affinity DataEC50: 38.4nMAssay Description:Topoisomerase I activity for single-strand breaks in the DNA substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Inhibition of topoisomerase-1 (unknown origin) using pBR 322 DNA as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Inhibitory effect on topoisomerase-I mediated DNA cleavage using supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:In vitro activity against topoisomerase-I mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Inhibition of topoisomerase-1 in human U251 cells assessed as inhibition of hypoxia-induced HIF-1alpha accumulation in nuclear extract after 6 to 24 ...More data for this Ligand-Target Pair