Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: >0nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0126nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0195nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: <0.100nMAssay Description:Modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aortic ring assessed as human urotensin-2 EC50 for induction of aortic ring contrac...More data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.160nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.290nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.340nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.398nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.450nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.540nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.540nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.631nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.661nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.724nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.760nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.813nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.830nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: 0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.09nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Antagonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as reduction in urotensin-2-induced contraction by measuring p...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as induction of contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.35nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.38nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aortic ring assessed as human urotensin-2 pEC50 for induction of aortic ring contra...More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aortic ring assessed as human urotensin-2 EC50 for induction of aortic ring contrac...More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at rat urotensin 2 receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Antagonist activity at UT2 receptor in Sprague-Dawley rat thoracic aorta ring assessed as pEC50 for hU2-induced aortic contractions at 10'-5M relativ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Mobilization of intracellular calcium in CHO cells transiently transfected with human Urotensin 2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Mobilization of intracellular calcium in CHO cells transiently transfected with human Urotensin 2 receptorMore data for this Ligand-Target Pair